Warnings
Cardiovascular risks - monitor BP and HR
Psychiatric effects possible
Serotonin syndrome risk with SSRIs
Not FDA approved
Phase III trials ongoing
Contraindications
MAO InhibitorsUncontrolled HypertensionCardiovascular DiseaseHyperthyroidismGlaucomaPregnancyBreastfeeding
Drug Interactions
MAOIsSSRIsSNRIsStimulantsSympathomimeticsCYP3A4 Inhibitors
Possible Side Effects
Dry MouthConstipationInsomniaIncreased Heart RateElevated Blood PressureMood Changes
Legal & Regulatory
FDA Status Not FDA Approved
WADA Status Prohibited in Sport
Prescription Required
Pregnancy
Category X - Contraindicated