Warnings
Not FDA approved
Monitor glucose levels
QT prolongation risk
Contraindications
PregnancyBreastfeedingSevere Hepatic Impairment
Drug Interactions
CYP3A4 InhibitorsCYP3A4 Inducers
Possible Side Effects
Peripheral EdemaIncreased Blood GlucoseQTc ProlongationConstipation
Legal & Regulatory
FDA Status Not FDA Approved
WADA Status Prohibited in Sport
Approved In Japan
Prescription Required
Pregnancy
Category X - Contraindicated