Dosing Protocol
Typical Dose 1.5 mg
Range 1 - 2 mg
Maintenance 1 mg daily
Cycle 8w on / 8w off
Pharmacokinetics
Half-Life 45 min
Onset 10 min
Peak 15 min
Duration 3.0 hrs
Bioavailability 90%
Primary Route Subcutaneous
Administration
Routes Subcutaneous, Topical
Injection Sites Abdomen, Thigh, Deltoid
Needle Gauge 29-31G
Syringe Type Insulin
Timing Morning, Evening
Reconstitution
Diluent Bacteriostatic Water
Volume 3 mL
Concentration 16667 mcg/mL
Stability 30 days refrigerated
Vial Sizes 50 mg
Special Instructions
Also available as topical cream (2-10% concentration). Cycle 8-12 weeks on, equal time off to maintain receptor sensitivity.